Current Medicinal Chemistry |
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5-HT receptors 5-HT1DB receptor activity of streptonigrin adenine adenosine AdoMet AdoMetDC agents Almotriptan alniditan amino acid antagonist antimigraine drug Bentham Science Publishers binding affinity biological activity biosynthesis bipyridyl brain brucei carboxylic cells chelate clinical trials complexes of streptonigrin compounds coronary artery Current Medicinal Chemistry DFMO disease dose eletriptan enzyme functional gGAPDH glycolytic glycosomal high affinity human hydrogen bond inhibition inhibitor interaction involved ligands mammalian mechanism Medicinal Chemistry melarsoprol metabolism metal complexes metal ions migraine migraine attacks moiety molecule Naratriptan neurogenic neurotensin non-peptidic NT analogs NT receptor parasite pathway peptide polyamine potency protein purine rational drug design reaction receptor subtype redox reported residue rhodesiense rizatriptan selectivity semiquinone sequence side chain sleeping sickness species spermidine streptonigrin structure studies substituted substrate suggested sumatriptan synthesis synthetase Table target treatment of migraine trigeminal trypanosomes trypanothione vitro Zn2+ Zolmitriptan