Current Medicinal Chemistry |
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2D NOESY Affinities and Selectivity amine amino acids analogs antagonist anthracycline antibiotics anticancer drugs antidepressant antipsychotic antisense aromatic atypical antipsychotic bacterial base pair Bentham Science Publishers brofaromine calicheamicin cells cisplatin clinical clozapine complex compounds covalent crosspeak D2-like D4 affinity D4 over D2 derivatives DNA duplex dopamine D4 receptors duplex duplex DNA enzyme flavin genes H3CO haloperidol hydrogen bond IC50 MAO inactivators inhibit MAO inhibitors of MAO interactions ligands linear prediction lipophilic MAO A inhibitors MAOA MAOIs mechanism Medicinal Chemistry membrane minor groove moiety molecules monoamine oxidase mRNA neuroleptics NMR spectroscopy NOESY NOESY data NOESY spectra nuclear DNA nucleic acid OCH3 Okazaki fragments oxazolidinones pathogens phenyl potential protein quinolones recent residues resistance reversible inhibitors reversible MAO ring role schizophrenia selectivity for dopamine sequence specific serotonin side effects strand structure studies substituted substrates synthesis target vancomycin vitro vivo