Current Medicinal Chemistry |
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0ssn 2-5A synthetase 2-5A trimer 2-5A-dependent RNase 3'-deoxyadenosine 3ncl ACAT inhibitory activity acid adenosine affinity agents alkyl amides amine amino anilide antagonist antisense artery wall baclofen barbiturates benzodiazepine benzodioxole binding catalytic catechol cells CH2Ph CH3 CH3 chimera cholesterol cholesterol-fed rats cholesteryl ester cleavage CLOGP CO2Et complex compounds cytochrome P450 decrease dependent RNase domain dose effect efficacy enzyme formation function GABA GABAA GABAB receptor IC50 value indolecarbazole inhibit ACAT inhibitor of PKC inhibits PKC inni0itos interaction inverse agonist isozymes ligands lipophilic MDMA mg/kg microsomes moiety molecule mouse mRNA nuclease nucleotide oligonucleotides oxidation partial agonist pharmacological phenyl picrotoxin plasma cholesterol potent ACAT inhibitors protein kinases rabbit reaction replaced ring SAR study selectivity sequence serine/threonine shown specific staurosporine substitution substrate subunit Table target tetrazole tn3t tni3 urea vitro vivo activity witn wnsn