Current Medicinal Chemistry |
Uobičajeni izrazi i fraze
3-substituent 7-dione A-ring a]benzimidazoles alkylation aminoglutethimide anticholinergic anticholinergic activity antitumor activity antitumor agents APBI apparent Kj Arimidex aromatase inhibitors atropine aziridine aziridine ring aziridinyl Bentham Science Publishers binding Bodor breast cancer Ca2+ channel cell lines cleavage clinical compounds correlation CQ resistance cytotoxicity drug design DT-diaphorase enzyme estrogen fadrazole herveline HuGrA HuGrB human granzyme hydrolysis hydrolytic hydroquinone iminoquinone inactivation inactive metabolite inhibition inhibitor of aromatase interactions irreversible inhibitors letrozole lipophilicity lymphocyte m/no-APBIs malaria mean graphs Medicinal Chemistry melanoma metabolic methatropine methscopolamine mg/kg IP Q7DX3,Day mydriatic nonsteroidal aromatase inhibitors nucleophile OVCAR-3 oxidation parasites PBI phosphodiesters PBI-A phosphate backbone potent anticholinergic propantheline protons pyrrolo[1,2-a]benzimidazole quinone quinone methide reaction reduced PBI reversal role serine protease shown in Chart soft analogs soft anticholinergics soft drugs steroid steroidal inhibitors strain structure studies substituent substrates synthetic Table target cell topoisomerase topoisomerase II toxicity treatment tryptase verapamil vitro vivo vorozole