Current Medicinal Chemistry |
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8-styrylxanthines active drug adenosine receptor ADEPT system affinity Aga adenosine receptor Aga antagonist Aga receptors Aga selectivity agents agonists alkyl amino antigen antitrypanosomal aromatic assays B-glu Batimastat Bentham Science Publishers binding biological activity carboxylic acid catalytic CH3 CH3 Chagas chemical chemotherapy cleavage co-workers collagen compound concentration conjugate CPG2 cruzi epimastigotes cruzi replication cytotoxicity derivatives disease dose doxorubicin effect enzyme ergosterol Fenoxycarb fibroblast fibroblast collagenase functional gelatinase gelatinase-A growth human hydroxamic acid infected inhibition values intracellular kcat Ketoconazole ligands mammalian host medicinal chemistry metalloproteinases MMP inhibitors moiety molecule neutrophil collagenase nitrogen mustard non-xanthine nude mice observed parasite peptides phosphinic phosphonic acids potent prodrug Prodrugs Cleaved protein rat brain ratio receptor subtypes residue solubility specific stromelysin structure studies substituent substrate synthesis Table Terbinafine tissues toxic triazole trypanosomes trypanothione trypomastigotes tumor values in nM vitro vivo xanthine xenografts zinc